Antibacterial steroidal alkaloids from Holarrhena antidysenteriaca

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摘要 Twonewsteroidalalkaloids,isoconkuressineandN-formylconessimine,togetherwith6knownsteroidalalkaloidsincludingconkuressine,conessine,isoconessimine,conimine,conarrhimine,andfuntudienine,wereisolatedfromtheseedsofHolarrhenaantidysenteriacaWall.exA.DC.Theirintrinsicantibacterialactivitiesandsynergisticeffectswithpenicillinandvancomycinwereanalyzedinmethicillinsensitivestaphylococcusaureus(MSSA)andmethicillinresistantstaphylococcusaureus(MRSA).Twoofthesteroidalalkaloidsincludingonenewcompound(N-formylconessimine)showedpotentialantibacterialactivityandpossessedsynergisticeffectswithpenicillinandvancomycin,respectively.
机构地区 不详
出版日期 2017年07月17日(中国期刊网平台首次上网日期,不代表论文的发表时间)
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